SCHEMBL7350408

SCHEMBL7350408

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2Cc3ccccc3C2)C1c1c[nH]c2ccccc12

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 1/20 0.69
CYP2C9 P11712 4/20 0.45
CYP1A2 P05177 3/20 0.45
ALDH1A1 P00352 2/20 0.45
CYP2D6 P10635 2/20 0.45
TSHR P16473 2/20 0.45
THPO P40225 2/20 0.45
PMP22 Q01453 2/20 0.44
GAA P10253 2/20 0.44
ADORA3 P0DMS8 3/20 0.43
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2C19 P33261 2/20 0.42
KMT2A Q03164 2/20 0.42
HIF1A Q16665 2/20 0.42
HSD17B10 Q99714 2/20 0.42
HPGD P15428 1/20 0.42
TP53 P04637 1/20 0.42
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7350735 0.83 PDE1C (0.69) PDE1CALDH1A1GAAADORA3HSD17B10
SCHEMBL7343547 0.83 ADORA3 (0.47) CYP2C9CYP1A2ALDH1A1CYP2D6TSHR
SCHEMBL7348023 0.83 CACNA1C (0.48) CYP2C9CYP1A2ALDH1A1CYP2D6TSHR
SCHEMBL7349519 0.83 ADORA3 (0.57) CYP2C9CYP1A2ALDH1A1CYP2D6TSHR
SCHEMBL7350412 0.81 PDE1C (0.65) PDE1CCYP2C9CYP1A2ALDH1A1CYP2D6
SCHEMBL10926541 0.81 PDE1C (0.57) PDE1CCYP2C9CYP1A2ALDH1A1CYP2D6
SCHEMBL7342397 0.81 ADORA3 (0.47) CYP2C9CYP1A2ALDH1A1CYP2D6TSHR
SCHEMBL7351367 0.80 ADORA3 (0.69) CYP2C9CYP1A2ALDH1A1CYP2D6TSHR
SCHEMBL7340139 0.79 ADORA3 (0.47) CYP2C9CYP1A2ALDH1A1CYP2D6TSHR
SCHEMBL10744164 0.78 ALDH1A1 (0.54) ALDH1A1TSHRGAAADORA3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed