SCHEMBL7344855

SCHEMBL7344855

O=C1N(CCCN2CCN(c3ccccc3)CC2)CCN1c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.63
DRD3 P35462 5/20 0.63
KCNH2 Q12809 1/20 0.59
HTR1A P08908 6/20 0.58
DRD5 P21918 1/20 0.55
CYP2D6 P10635 1/20 0.55
HTR7 P34969 2/20 0.54
SIGMAR1 Q99720 3/20 0.54
HTR2A P28223 2/20 0.53
HDAC1 Q13547 2/20 0.52
HRH1 P35367 1/20 0.51
TMEM97 Q5BJF2 1/20 0.51
ADRB2 P07550 1/20 0.51
CHRM2 P08172 1/20 0.51
CHRM4 P08173 1/20 0.51
ADRB1 P08588 1/20 0.51
CHRM5 P08912 1/20 0.51
CHRM1 P11229 1/20 0.51
CHRM3 P20309 1/20 0.51
DRD4 P21917 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7347501 0.99 DRD2 (0.62) DRD2DRD3KCNH2HTR1ADRD5
SCHEMBL7068893 0.97 KCNH2 (0.64) DRD2DRD3KCNH2HTR1ADRD5
SCHEMBL7346970 0.83 KCNH2 (0.67) DRD2DRD3KCNH2HTR1AHTR7
SCHEMBL9299310 0.81 DRD2 (0.54) DRD2DRD3KCNH2HTR1ASIGMAR1
SCHEMBL5988317 0.81 KCNH2 (0.88) DRD2DRD3KCNH2HTR1ACYP2D6
SCHEMBL7344989 0.81 HTR1A (0.64) DRD2DRD3HTR1ADRD5CYP2D6
SCHEMBL6924599 0.81 ADRA1A (0.57) DRD2DRD3HTR1AADRA1DADRA1A
SCHEMBL6924603 0.80 DRD3 (0.55) DRD2DRD3HTR1AHTR7
SCHEMBL8143460 0.80 HTR1A (0.61) DRD2HTR1AHTR2A
SCHEMBL7935881 0.79 DRD2 (0.61) DRD2DRD3KCNH2HTR2AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5281594-A Dopamine antagonist, Parkinson's disease and drug addiction THE UPJOHN COMPANY (US) 1994-01-25 US disclosed
EP-0536279-A1 SUBSTITUTED 1-(ALKOXYPHENYL)PIPERAZINES WITH CNS AND ANTIHYPERTENSIVE ACTIVITY THE UPJOHN COMPANY (US) 1993-04-14 EP disclosed
WO-1992000282-A1 SUBSTITUTED 1-(ALKOXYPHENYL)PIPERAZINES WITH CNS AND ANTIHYPERTENSIVE ACTIVITY THE UPJOHN COMPANY (US) 1992-01-09 WO disclosed