SCHEMBL7345087

SCHEMBL7345087

N=C(N)Nc1cccc(C(=O)NCC(=O)NC2(CCC(=O)O)C=CSC2)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.38
ITGB3 P05106 7/20 0.38
ITGA2B P08514 3/20 0.38
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
F10 P00742 2/20 0.36
PRSS1 P07477 1/20 0.36
ITGB1 P05556 4/20 0.35
ITGAV P06756 4/20 0.35
ITGA5 P08648 4/20 0.35
MDM4 O15151 3/20 0.35
MDM2 Q00987 3/20 0.35
EPHX2 P34913 2/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
GAA P10253 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7343247 0.91 EPHX2 (0.36) SMN1; SMN2F10PRSS1EPHX2MEN1
SCHEMBL7345104 0.88 ITGB3 (0.34) SMN1; SMN2ITGB3ITGA2BHTTL3MBTL1
SCHEMBL7343256 0.79 KMT2A (0.37) SMN1; SMN2ITGB3ITGAVEPHX2MEN1
SCHEMBL6773153 0.76 ITGB3 (0.55) SMN1; SMN2ITGB3ITGA2BHTTL3MBTL1
SCHEMBL7340450 0.76 HTT (0.37) SMN1; SMN2ITGB3ITGA2BHTTL3MBTL1
SCHEMBL6366986 0.74 PLA2G10 (0.47) SMN1; SMN2ITGB3ITGA2BHTTL3MBTL1
SCHEMBL27502754 0.74 ITGB3 (0.47) SMN1; SMN2ITGB3ITGA2BHTTL3MBTL1
Hydrochloric Acid SCHEMBL6773326 0.73 PLA2G10 (0.46) SMN1; SMN2ITGB3ITGA2BHTTL3MBTL1
Hydrochloric Acid SCHEMBL6368863 0.73 PLA2G10 (0.46) SMN1; SMN2ITGB3ITGA2BHTTL3MBTL1
SCHEMBL7348597 0.73 ITGB3 (0.38) SMN1; SMN2ITGB3ITGA2BHTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed