SCHEMBL7345620

SCHEMBL7345620

CCCCS(=O)(=O)N[C@@H](Cc1ccc(OCCCC(=O)OCC)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 11/20 0.56
ITGA2B P08514 11/20 0.56
ITGAV P06756 1/20 0.53
CHRM2 P08172 1/20 0.53
SLC6A4 P31645 1/20 0.53
LTA4H P09960 4/20 0.42
MAPT P10636 1/20 0.41
ACACB O00763 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352181 0.90 ITGB3 (0.61) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7342244 0.88 ITGB3 (0.62) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7350681 0.85 ITGB3 (0.52) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7348077 0.85 ITGB3 (0.54) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7351394 0.84 MAPT (0.44) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL6873358 0.84 TDP1 (0.46) ITGB3ITGA2BITGAVLTA4H
SCHEMBL7351843 0.82 ITGB3 (0.43) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7297528 0.79 ITGB3 (0.58) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7464600 0.78 ITGB3 (0.48) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL6286612 0.78 LTA4H (0.47) ITGB3ITGA2BLTA4HMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907637-A1 PHENYLALAMINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 1999-04-14 EP disclosed
WO-1998000395-A1 PHENYLALAMINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 1998-01-08 WO disclosed