SCHEMBL7350681

SCHEMBL7350681

CCCCS(=O)(=O)N[C@@H](Cc1ccc(OCCCC(=O)CN=NO)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 17/20 0.52
ITGA2B P08514 17/20 0.52
ITGAV P06756 1/20 0.49
CHRM2 P08172 1/20 0.49
SLC6A4 P31645 1/20 0.49
NPR3 P17342 1/20 0.37
ACACB O00763 1/20 0.36
BCL2 P10415 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352181 0.86 ITGB3 (0.61) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7345620 0.85 ITGB3 (0.56) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7342244 0.84 ITGB3 (0.62) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7348077 0.81 ITGB3 (0.54) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7407517 0.77 ITGB3 (0.50) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7297528 0.76 ITGB3 (0.58) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL8720830 0.74 ITGB3 (0.59) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL8722904 0.74 ITGB3 (0.59) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7280760 0.73 ITGB3 (0.62) ITGB3ITGA2BITGAVCHRM2SLC6A4
SCHEMBL7351394 0.71 MAPT (0.44) ITGB3ITGA2BITGAVCHRM2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0907637-A1 PHENYLALAMINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 1999-04-14 EP disclosed
WO-1998000395-A1 PHENYLALAMINE DERIVATIVES AS INTEGRIN INHIBITORS MERCK PATENT GMBH (DE) 1998-01-08 WO disclosed