SCHEMBL7345812

SCHEMBL7345812

N=C(N)Nc1ccccc1C(=O)NCC(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.47
KEAP1 Q14145 1/20 0.47
PPARG P37231 3/20 0.46
MAPT P10636 1/20 0.46
ITGB3 P05106 2/20 0.44
ITGB1 P05556 1/20 0.44
ITGAV P06756 1/20 0.44
ITGA5 P08648 1/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HTT P42858 1/20 0.44
NR1H4 Q96RI1 1/20 0.42
PDCD1 Q15116 1/20 0.42
CD274 Q9NZQ7 1/20 0.42
EGLN1 Q9GZT9 1/20 0.42
ITGA2B P08514 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MT-CO2 P00403 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27419805 0.89 BACE1 (0.50) BACE1KEAP1PPARGMAPTITGB3
SCHEMBL21800978 0.81 CYP2C19 (0.58) BACE1KEAP1MAPTITGB3ITGB1
SCHEMBL13992226 0.81 BACE1 (0.68) BACE1PPARGMAPTMEN1KMT2A
SCHEMBL4952951 0.79 LMNA (0.63) BACE1PPARGMAPTKDM4EALDH1A1
SCHEMBL233797 0.79 KMT2A (0.57) MAPTKDM4EALDH1A1MEN1KMT2A
Benzene SCHEMBL27690342 0.79 KMT2A (0.57) MAPTKDM4EALDH1A1MEN1KMT2A
SCHEMBL31448014 0.78 KEAP1 (0.62) KEAP1MAPTKDM4EKMT2AHTT
SCHEMBL9302237 0.78 F10 (0.49) MAPTKDM4EALDH1A1MEN1KMT2A
SCHEMBL8768375 0.78 HPGD (0.51) BACE1KEAP1PPARGMAPTITGB3
SCHEMBL17087190 0.78 KEAP1 (0.51) BACE1KEAP1PPARGMAPTITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP disclosed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO disclosed