SCHEMBL7345846

SCHEMBL7345846

CCOC(=O)CCC1=CC(Cl)=CC(Cl)(NC(=O)CNC(=O)c2cccc(NC3=NCC(C)(C)CN3)c2)C1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.38
ITGAV P06756 19/20 0.38
ITGB6 P18564 12/20 0.38
ITGB1 P05556 1/20 0.38
ITGA5 P08648 1/20 0.38
ITGB5 P18084 1/20 0.38
ITGB8 P26012 1/20 0.38
ITGA8 P53708 1/20 0.38
HTR1A P08908 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR7 P34969 1/20 0.34
HTR2B P41595 1/20 0.34
HTR5A P47898 1/20 0.34
HTR6 P50406 1/20 0.34
ITGA2B P08514 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348218 0.80 NAMPT (0.51)
SCHEMBL7367300 0.80 ITGB3 (0.51) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7343122 0.79 NAMPT (0.42)
SCHEMBL7345255 0.79 ITGB3 (0.53) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7340484 0.79 ALDH1A1 (0.34) ITGB1ITGA5
SCHEMBL7340476 0.79 ALDH1A1 (0.34) ITGB1ITGA5
SCHEMBL7836124 0.75 ITGB3 (0.52) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7346226 0.74 LMNA (0.35) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7836126 0.73 ITGB3 (0.48) ITGB3ITGAVITGB6ITGB1ITGA5
SCHEMBL7343261 0.72 ITGB3 (0.40) ITGB3ITGAVITGB6ITGB1ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP disclosed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO disclosed