SCHEMBL7346229

SCHEMBL7346229

N=C(N)Nc1cccc(C(=O)NCC(=O)NC2(Br)C=C(Cl)C=C(CCC(=O)O)C2O)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 8/20 0.36
ITGA2B P08514 3/20 0.36
F10 P00742 2/20 0.35
PRSS1 P07477 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GAA P10253 1/20 0.33
ITGAV P06756 6/20 0.32
ITGB6 P18564 3/20 0.32
EPHX2 P34913 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ITGB1 P05556 1/20 0.32
ITGB5 P18084 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7346234 0.89 KMT2A (0.34) ITGB3ITGA2BF10PRSS1MAPT
SCHEMBL7375174 0.82 ITGB3 (0.33) ITGB3ITGA2BITGAVITGB6
SCHEMBL7340934 0.81 ITGB3 (0.37) ITGB3ITGA2BF10PRSS1SMN1; SMN2
SCHEMBL7336943 0.80 NPC1 (0.33) ITGB3ITGA2BSMN1; SMN2LMNAL3MBTL1
SCHEMBL7343452 0.76 ITGB3 (0.37) ITGB3ITGA2BF10PRSS1SMN1; SMN2
SCHEMBL7348225 0.75 ITGB3 (0.38) ITGB3ITGA2BF10PRSS1SMN1; SMN2
SCHEMBL7341549 0.75
SCHEMBL7348823 0.75 ITGB3 (0.37) ITGB3ITGA2BF10PRSS1SMN1; SMN2
SCHEMBL7347196 0.74 HTT (0.37) ITGB3ITGA2BF10PRSS1SMN1; SMN2
SCHEMBL7341117 0.74 ITGB3 (0.39) ITGB3ITGA2BF10PRSS1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed