SCHEMBL7346358

SCHEMBL7346358

CN1CCN(CC(=O)N(c2ccccc2)c2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.62
CACNA2D1 P54289 5/20 0.52
CACNA1B Q00975 5/20 0.52
CACNB1 Q02641 5/20 0.52
CACNA1C Q13936 5/20 0.52
POLB P06746 1/20 0.49
HTT P42858 2/20 0.48
LMNA P02545 2/20 0.47
TP53 P04637 1/20 0.47
KMT2A Q03164 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
MEN1 O00255 1/20 0.46
CRHBP P24387 1/20 0.46
ATM Q13315 1/20 0.46
CRHR2 Q13324 1/20 0.46
TLR9 Q9NR96 1/20 0.46
SIRT6 Q8N6T7 1/20 0.45
HTR1A P08908 1/20 0.45
TSHR P16473 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339023 0.87 CACNA2D1 (0.65) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL1361808 0.84 ALDH1A1 (0.50) ALDH1A1HTTLMNAKMT2AL3MBTL1
SCHEMBL7339537 0.82 CACNA2D1 (0.56) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1C
Hydrochloric Acid SCHEMBL7341072 0.81 CACNA2D1 (0.53) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL17147663 0.81 ALDH1A1 (0.47) ALDH1A1POLBHTTLMNAKMT2A
SCHEMBL7342475 0.80 CACNA2D1 (0.54) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL27959322 0.80 CHRM2 (0.47) ALDH1A1HTTLMNAKMT2ASIRT6
SCHEMBL7346027 0.79 CACNA2D1 (0.53) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL7339671 0.79 CACNA2D1 (0.53) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL7342378 0.78 CACNA2D1 (0.52) ALDH1A1CACNA2D1CACNA1BCACNB1CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0658157-A1 DIARYL PIPERAZINOACETAMIDE COMPOUNDS AS ANTIMUSCARINIC AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-06-21 EP disclosed
WO-1994005648-A1 DIARYL PIPERAZINOACETAMIDE COMPOUNDS AS ANTIMUSCARINIC AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-17 WO disclosed
EP-0585500-A1 Diaryl piperazineacetamides as antimuscarinic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1994-03-09 EP disclosed