SCHEMBL7347205

SCHEMBL7347205

CC(C[O])CS(=O)(=O)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.54
MMP13 P45452 2/20 0.45
MMP1 P03956 1/20 0.45
HSD11B1 P28845 6/20 0.43
POLB P06746 1/20 0.42
ALDH1A1 P00352 3/20 0.41
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.40
CYP2C19 P33261 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HTR6 P50406 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2444476 0.84 PSIP1 (0.59) PSIP1MMP13MMP1HSD11B1POLB
SCHEMBL7347214 0.82 PSIP1 (0.52) PSIP1MMP13MMP1HSD11B1POLB
SCHEMBL778303 0.81 PSIP1 (0.60) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL12249321 0.81 PSIP1 (0.50) PSIP1MMP13MMP1HSD11B1ALDH1A1
SCHEMBL20780856 0.81 PSIP1 (0.55) PSIP1MMP13MMP1HSD11B1POLB
SCHEMBL4680931 0.81 MMP13 (0.42) PSIP1MMP13MMP1ALDH1A1HTT
SCHEMBL15214393 0.81 PSIP1 (0.50) PSIP1MMP13MMP1HSD11B1POLB
SCHEMBL6098280 0.79 PSIP1 (0.48) PSIP1MMP13MMP1HSD11B1POLB
SCHEMBL4682741 0.79 NAPRT (0.47) MMP13MMP1POLBHSD17B10
SCHEMBL25015902 0.78 PSIP1 (0.52) PSIP1MMP13MMP1HSD11B1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed