SCHEMBL7348556

SCHEMBL7348556

CC(NS(=O)(=O)CC(N)=O)(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
MAPT P10636 1/20 0.44
CYP2C19 P33261 2/20 0.40
NR3C2 P08235 1/20 0.40
KCNN4 O15554 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD11B1 P28845 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
RECQL P46063 2/20 0.37
ALDH1A1 P00352 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7304270 0.84 KCNN4 (0.43) KMT2AMAPTCYP2C19NR3C2KCNN4
SCHEMBL7301814 0.80 KMT2A (0.40) KMT2AMAPTHSD11B1ALDH1A1F2
SCHEMBL21393560 0.73 ALDH1A1 (0.38) MAPTALDH1A1NPC1
SCHEMBL4401320 0.70 CA1 (0.50) KMT2AMAPTNR3C2ALDH1A1MEN1
SCHEMBL7315311 0.70 MAPT (0.43) KMT2AMAPTCYP2C19HIF1AHSD11B1
SCHEMBL28376940 0.70 MAPT (0.55) KMT2AMAPTCYP2C19NR3C2KCNN4
SCHEMBL28710857 0.67 MAPT (0.52) KMT2AMAPTCYP2C19KCNN4HIF1A
SCHEMBL168185 0.67 MAPT (0.44) KMT2AMAPTCYP2C19NR3C2HIF1A
SCHEMBL4557719 0.67 CYP2C19 (0.43) CYP2C19HSD11B1CYP1A2MAPK1
SCHEMBL5674843 0.67 MAPT (0.52) KMT2AMAPTCYP2C19NR3C2KCNN4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0931788-B1 Metalloprotease inhibitors PFIZER LTD (GB) 2002-11-06 EP disclosed
US-6090852-A MATRIX METALLOPROTEASE INHIBITOR PFIZER INC (US) 2000-07-18 US disclosed
EP-0931788-A2 Metalloprotease inhibitors Pfizer Limited (GB) 1999-07-28 EP disclosed