SCHEMBL7315311

SCHEMBL7315311

CN(C(C)(c1ccccc1)c1ccccc1)S(=O)(=O)CC(N)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD11B1 P28845 2/20 0.41
CYP2C19 P33261 2/20 0.39
HIF1A Q16665 1/20 0.39
ESR2 Q92731 1/20 0.37
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
RECQL P46063 1/20 0.36
RAB9A P51151 1/20 0.36
OPRM1 P35372 2/20 0.36
DRD3 P35462 2/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
SLC22A2 O15244 1/20 0.35
SLC22A1 O15245 1/20 0.35
PGR P06401 1/20 0.35
THRB P10828 1/20 0.35
ADRB3 P13945 1/20 0.35
OPRK1 P41145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7309339 0.87 CYP2C19 (0.44) MAPTKMT2AHSD11B1CYP2C19HIF1A
SCHEMBL7313045 0.78 HSD11B1 (0.39) MAPTKMT2AHSD11B1ALDH1A1
SCHEMBL7479619 0.74 ALDH1A1 (0.33) ALDH1A1
SCHEMBL7478269 0.71 MMP3 (0.57) KMT2AALDH1A1NPC1RAB9ATSHR
SCHEMBL7348556 0.70 KMT2A (0.44) MAPTKMT2AHSD11B1CYP2C19HIF1A
SCHEMBL7306332 0.70 CYP2C19 (0.41) MAPTKMT2AHSD11B1CYP2C19ALDH1A1
SCHEMBL7302947 0.69 MMP3 (0.59) KMT2ANPC1RAB9ATSHRTDP1
SCHEMBL6245112 0.66 ALDH1A1 (0.42) MAPTKMT2AALDH1A1TSHR
SCHEMBL2813766 0.65 MAPT (0.55) MAPTKMT2ACYP2C19HIF1AALDH1A1
SCHEMBL362442 0.65 KMT2A (0.55) MAPTKMT2ACYP2C19HIF1AESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0931788-B1 Metalloprotease inhibitors PFIZER LTD (GB) 2002-11-06 EP disclosed
US-6090852-A MATRIX METALLOPROTEASE INHIBITOR PFIZER INC (US) 2000-07-18 US disclosed
EP-0931788-A2 Metalloprotease inhibitors Pfizer Limited (GB) 1999-07-28 EP disclosed