SCHEMBL7349883

SCHEMBL7349883

COc1cc(OC[C]=O)ccc1NC(C)=O

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
HSD17B1 P14061 1/20 0.54
HSD17B2 P37059 1/20 0.54
MAPT P10636 3/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
PKM P14618 1/20 0.51
GAA P10253 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
PTK2 Q05397 1/20 0.48
CYP1A1 P04798 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP1B1 Q16678 1/20 0.48
HPGD P15428 2/20 0.47
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
LMNA P02545 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5657703 0.84 ALDH1A1 (0.66) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL2191052 0.82 HSD17B1 (0.75) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL30622065 0.82 HSD17B1 (0.75) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL2641220 0.77 CA2 (0.55) ALDH1A1GAANPC1CYP1A2LMNA
SCHEMBL6975514 0.75 TP53 (0.56) ALDH1A1MAPTMEN1KMT2APKM
SCHEMBL5259715 0.75 BRD4 (0.63) ALDH1A1MAPTMEN1KMT2AGAA
SCHEMBL10789373 0.75 TDP1 (0.58) ALDH1A1MAPTMEN1KMT2AGAA
SCHEMBL14384842 0.74 MEN1 (0.62) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL30615269 0.74 HSD17B1 (0.57) ALDH1A1HSD17B1HSD17B2MAPTMEN1
SCHEMBL7356599 0.74 KMT2A (0.67) ALDH1A1MAPTMEN1KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5985869-A USEFUL AS VASODILATORS, HYPOTENSIVE AGENTS, WATER DIURETICS, PLATELET AGGLUTINATION INHIBITORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1999-11-16 US disclosed
US-5753677-A Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5559230-A VASOPRESSIN ANTAGONISTS, QUINOLINES, BENZAZEPINES, VASODILATION, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-09-24 US disclosed
EP-0450097-B1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
WO-1991005549-A1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-05-02 WO disclosed