SCHEMBL7350667

SCHEMBL7350667

CN/C(=N\C#N)Nc1cccc(C(=O)NCC(=O)Nc2ccccc2CCC(=O)O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.44
KCNK9 Q9NPC2 1/20 0.44
ITGB1 P05556 1/20 0.43
ITGA5 P08648 1/20 0.43
HTT P42858 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MAPT P10636 2/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 2/20 0.38
ALDH1A1 P00352 3/20 0.37
NPSR1 Q6W5P4 1/20 0.37
GPR139 Q6DWJ6 1/20 0.37
BCHE P06276 1/20 0.37
SENP1 Q9P0U3 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
RXFP1 Q9HBX9 1/20 0.36
CASP6 P55212 1/20 0.36
MCL1 Q07820 1/20 0.36
CTDSP1 Q9GZU7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7350687 1.00 KCNK3 (0.44) KCNK3KCNK9ITGB1ITGA5HTT
SCHEMBL7345956 0.92 KCNK3 (0.45) KCNK3KCNK9ITGB1ITGA5HTT
SCHEMBL7346968 0.92 KCNK3 (0.45) KCNK3KCNK9ITGB1ITGA5HTT
SCHEMBL7338973 0.90 SENP1 (0.46) KCNK3KCNK9ITGB1ITGA5HTT
SCHEMBL7338982 0.90 SENP1 (0.46) KCNK3KCNK9ITGB1ITGA5HTT
SCHEMBL7383610 0.81 KCNK3 (0.48) KCNK3KCNK9L3MBTL1MAPTSMN1; SMN2
SCHEMBL7383607 0.81 KCNK3 (0.48) KCNK3KCNK9L3MBTL1MAPTSMN1; SMN2
SCHEMBL6777356 0.80 ITGB1 (0.42) ITGB1ITGA5HTTL3MBTL1SMN1; SMN2
SCHEMBL7350678 0.79 ITGB1 (0.53) ITGB1ITGA5LMNAGPR139
SCHEMBL6779632 0.78 GPR139 (0.48) ITGB1ITGA5GPR139MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850221-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1998-07-01 EP claimed
WO-1997008145-A1 META-GUANIDINE, UREA, THIOUREA OR AZACYCLIC AMINO BENZOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-03-06 WO claimed