SCHEMBL7350735

SCHEMBL7350735

COC(=O)C1=C(C)NC(C)=C(C(=O)OCCN2C(=O)c3ccccc3C2=O)C1c1c[nH]c2ccccc12

nearest known ligand 0.69

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 1/20 0.69
HSD17B10 Q99714 3/20 0.62
ALDH1A1 P00352 2/20 0.48
PKM P14618 1/20 0.48
HPGD P15428 2/20 0.45
MAPK1 P28482 1/20 0.45
GAA P10253 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ADORA3 P0DMS8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7350408 0.83 PDE1C (0.69) PDE1CHSD17B10ALDH1A1HPGDGAA
SCHEMBL7342557 0.83 HSD17B10 (0.66) HSD17B10ALDH1A1HPGDMAPK1GAA
SCHEMBL7344861 0.83 HSD17B10 (0.66) HSD17B10ALDH1A1HPGDMAPK1GAA
SCHEMBL7348263 0.83 HSD17B10 (0.66) HSD17B10ALDH1A1HPGDGAASMN1; SMN2
SCHEMBL7344176 0.81 HSD17B10 (0.66) HSD17B10ALDH1A1PKMHPGDMAPK1
SCHEMBL9673018 0.80 CYP2C9 (0.68) HSD17B10ALDH1A1HPGDGAASMN1; SMN2
SCHEMBL7347242 0.80 ADORA3 (0.69) HSD17B10ALDH1A1HPGDMAPK1SMN1; SMN2
SCHEMBL7343943 0.79 HSD17B10 (0.66) HSD17B10ALDH1A1PKMHPGDMAPK1
SCHEMBL7340301 0.78 HSD17B10 (0.67) HSD17B10ALDH1A1HPGDMAPK1GAA
SCHEMBL7341261 0.78 KDM4E (0.67) HSD17B10ALDH1A1HPGDGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4833150-A HYPOTENSIVES, ANTIARRHYTHMIA AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1989-05-23 US disclosed
US-4652573-A HYPOTENSIVE AGENTS NELSON RESEARCH & DEVELOPMENT CO. (US) 1987-03-24 US disclosed
EP-0194685-A1 1,4-Dihydropyridines Whitby Research Incorporated (US) 1986-09-17 EP disclosed