SCHEMBL7352170

SCHEMBL7352170

CC(C)CCC(NC(=O)NC(C)(C)C)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@H](CC(N)=O)NS(=O)(=O)C=Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.39
CYP3A4 P08684 3/20 0.39
LMNA P02545 2/20 0.39
USP2 O75604 1/20 0.39
CYP2D6 P10635 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
HIF1A Q16665 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
POLB P06746 1/20 0.38
ABCC3 O15438 1/20 0.38
ABCC4 O15439 1/20 0.38
CACNA1F O60840 1/20 0.38
ABCB11 O95342 1/20 0.38
ABCB1 P08183 1/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
TACR2 P21452 1/20 0.38
TBXAS1 P24557 1/20 0.38
OPRM1 P35372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352165 1.00 GAA (0.39) GAACYP3A4LMNAUSP2CYP2D6
SCHEMBL7424747 0.90 HTT (0.46) GAAPOLBADAM17HTTREN
SCHEMBL7424741 0.90 HTT (0.46) GAAPOLBADAM17HTTREN
SCHEMBL7358901 0.88 CYP3A4 (0.41) CYP3A4LMNAUSP2CYP2D6ALDH1A1
SCHEMBL7353045 0.87 ADAM17 (0.44) GAAPOLBADAM17HTTPSEN1
SCHEMBL7353051 0.87 ADAM17 (0.44) GAAPOLBADAM17HTTPSEN1
SCHEMBL7358269 0.85 CYP3A4 (0.39) CYP3A4LMNAUSP2CYP2D6ALDH1A1
SCHEMBL7360300 0.81 BACE1 (0.40) CYP3A4ABCC3ABCC4CACNA1FABCB11
SCHEMBL8897548 0.77 BACE1 (0.33) CYP3A4ALDH1A1ADAM17HTTREN
SCHEMBL8897311 0.75 REN (0.38) ALDH1A1REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614522-A SULFONAMIDE AND UREA-CONTAINING HYDROXYETHYLAMINE COMPOUNDS G.D. SEARLE & CO. (US) 1997-03-25 US disclosed
EP-0558673-A1 RETROVIRAL PROTEASE INHIBITORS. MONSANTO CO (US) 1993-09-08 EP disclosed
WO-1992008699-A1 RETROVIRAL PROTEASE INHIBITORS MONSANTO COMPANY (US) 1992-05-29 WO disclosed