SCHEMBL8897548

SCHEMBL8897548

CC(C)CCC(NC(=O)NC(C)(C)C)[C@H](O)[C@H](Cc1ccccc1)NC(=O)CN(C(C)(C)C)S(=O)(=O)/C=C/c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.33
REN P00797 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
EGFR P00533 1/20 0.31
CTSD P07339 1/20 0.31
SPPL2A Q8TCT8 1/20 0.31
ADAM17 P78536 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360719 0.87 BACE1 (0.36) BACE1RENCTSDSPPL2A
SCHEMBL8899924 0.84 BACE1 (0.36) BACE1RENCTSD
SCHEMBL7353583 0.83 BACE1 (0.37) BACE1RENCTSD
SCHEMBL7424741 0.82 HTT (0.46) RENHTTADAM17
SCHEMBL7424747 0.82 HTT (0.46) RENHTTADAM17
SCHEMBL7476233 0.81 SPPL2A (0.38) BACE1CTSDSPPL2A
SCHEMBL7353051 0.80 ADAM17 (0.44) HTTCTSDADAM17
SCHEMBL7353045 0.80 ADAM17 (0.44) HTTCTSDADAM17
SCHEMBL8606263 0.77 BACE1 (0.35) BACE1RENALDH1A1
SCHEMBL7352170 0.77 GAA (0.39) BACE1RENALDH1A1CYP3A4HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5614522-A SULFONAMIDE AND UREA-CONTAINING HYDROXYETHYLAMINE COMPOUNDS G.D. SEARLE & CO. (US) 1997-03-25 US disclosed