SCHEMBL7352452

SCHEMBL7352452

CCCc1[nH]c2ccc(NS(=O)(=O)c3cccc4cccnc34)cc2c1C(=O)CCc1ccc(C#N)cc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
LMNA P02545 1/20 0.44
PKLR P30613 4/20 0.44
HTR6 P50406 1/20 0.43
TRPV1 Q8NER1 1/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
FABP1 P07148 2/20 0.41
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
GAA P10253 1/20 0.41
BRD4 O60885 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
PKM P14618 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357627 0.80 PKLR (0.46) ALDH1A1LMNAPKLRTRPV1MEN1
SCHEMBL7353803 0.79 PKLR (0.47) ALDH1A1LMNAPKLRHTR6MEN1
SCHEMBL7356136 0.79 ALDH1A1 (0.48) ALDH1A1LMNAPKLRHTR6MEN1
SCHEMBL8524454 0.73 PKLR (0.49) ALDH1A1LMNAPKLRMEN1KMT2A
SCHEMBL7352541 0.73 PKLR (0.48) ALDH1A1LMNAPKLRHTR6MEN1
SCHEMBL7356024 0.72 F2 (0.47) ALDH1A1TP53HTTPKM
SCHEMBL6572882 0.71 MEN1 (0.52) ALDH1A1PKLRMEN1KMT2AFABP1
SCHEMBL8525044 0.71 PKLR (0.49) ALDH1A1PKLRMEN1KMT2AFABP1
SCHEMBL6633872 0.71 F2 (0.50) ALDH1A1PKLRMEN1KMT2ATP53
SCHEMBL7358688 0.70 PKLR (0.47) ALDH1A1LMNAPKLRHTR6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed