SCHEMBL7357627

SCHEMBL7357627

CCn1cc(C(=O)CCc2ccc(C#N)cc2)c2cc(NS(=O)(=O)c3cccc4cccnc34)ccc21

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PKLR P30613 5/20 0.46
NTSR1 P30989 2/20 0.46
F2 P00734 1/20 0.44
ALDH1A1 P00352 3/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
FABP1 P07148 2/20 0.42
TP53 P04637 1/20 0.42
HTT P42858 1/20 0.42
GAA P10253 1/20 0.42
SLC2A1 P11166 2/20 0.41
LMNA P02545 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
BRD4 O60885 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7353803 0.92 PKLR (0.47) PKLRNTSR1F2ALDH1A1MEN1
SCHEMBL7352541 0.84 PKLR (0.48) PKLRNTSR1F2ALDH1A1MEN1
SCHEMBL7354601 0.83 F2 (0.59) PKLRNTSR1F2ALDH1A1MEN1
SCHEMBL7354443 0.80 PKLR (0.47) PKLRNTSR1F2ALDH1A1MEN1
SCHEMBL7352452 0.80 ALDH1A1 (0.44) PKLRALDH1A1MEN1KMT2AFABP1
SCHEMBL7358688 0.80 PKLR (0.47) PKLRNTSR1F2ALDH1A1MEN1
SCHEMBL6633872 0.76 F2 (0.50) PKLRNTSR1F2ALDH1A1MEN1
SCHEMBL8524454 0.75 PKLR (0.49) PKLRALDH1A1MEN1KMT2AFABP1
SCHEMBL7358689 0.75 NTSR1 (0.67) PKLRNTSR1ALDH1A1MEN1KMT2A
SCHEMBL7357042 0.74 MAPT (0.43) ALDH1A1TP53GAALMNAHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed