SCHEMBL8524454

SCHEMBL8524454

N#Cc1ccc(CNC(=O)c2cccc3ccc(NS(=O)(=O)c4cccc5cccnc45)cc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKLR P30613 4/20 0.49
MEN1 O00255 5/20 0.49
KMT2A Q03164 5/20 0.49
EGLN1 Q9GZT9 4/20 0.48
ALDH1A1 P00352 3/20 0.48
GAA P10253 1/20 0.48
FABP1 P07148 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
LMNA P02545 1/20 0.44
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8525044 0.94 PKLR (0.49) PKLRMEN1KMT2AEGLN1ALDH1A1
Hydrochloric Acid SCHEMBL8524038 0.87 F2 (0.56) PKLRMEN1KMT2AALDH1A1GAA
SCHEMBL7358688 0.87 PKLR (0.47) PKLRMEN1KMT2AEGLN1ALDH1A1
SCHEMBL8524665 0.84 SLC16A3 (0.42) PKLRMEN1KMT2AEGLN1ALDH1A1
SCHEMBL8525755 0.82 HSP90AA1 (0.49)
Hydrochloric Acid SCHEMBL8525302 0.82 F2 (0.56) PKLRMEN1KMT2AALDH1A1GAA
SCHEMBL8525757 0.82 KMT2A (0.44) PKLRMEN1KMT2AEGLN1ALDH1A1
SCHEMBL8525447 0.81 PKLR (0.44) PKLR
SCHEMBL7352541 0.77 PKLR (0.48) PKLRMEN1KMT2AALDH1A1GAA
SCHEMBL7353803 0.76 PKLR (0.47) PKLRMEN1KMT2AALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999029670-A2 AMINOCARBONYLTETRALIN AND DIHYDRONAPHTALENE DERIVATES AS THROMBIN INHIBITORS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-17 WO disclosed