SCHEMBL7353058

SCHEMBL7353058

CC(Nc1c(N)ccc2ccccc12)P(=O)(O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.44
CA2 P00918 1/20 0.44
MMP2 P08253 1/20 0.44
MMP9 P14780 1/20 0.44
MMP8 P22894 1/20 0.44
MMP14 P50281 1/20 0.44
CA14 Q9ULX7 1/20 0.44
FDPS P14324 1/20 0.40
ACP3 P15309 4/20 0.37
KCNJ11 Q14654 3/20 0.36
CMA1 P23946 3/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ANPEP P15144 1/20 0.35
G6PD P11413 1/20 0.35
NCEH1 Q6PIU2 1/20 0.35
CTSG P08311 1/20 0.35
HCRTR1 O43613 1/20 0.35
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7358348 0.81 ALDH1A1 (0.43) CA12CA2MMP2MMP9MMP8
SCHEMBL7357998 0.79 CA12 (0.48) CA12CA2MMP2MMP9MMP8
SCHEMBL680370 0.78 AKR1B1 (0.40) KCNJ11NPC1RAB9AKDM4EG6PD
SCHEMBL7355497 0.76 ACP3 (0.42) CA12CA2MMP2MMP9MMP8
SCHEMBL4430656 0.75 CA12 (0.71) CA12CA2MMP2MMP9MMP8
SCHEMBL8621279 0.73 ALDH1A1 (0.36) CA2KCNJ11RAB9AKDM4EG6PD
SCHEMBL21555507 0.70 ALDH1A1 (0.46) NPC1RAB9AKDM4EG6PDNCEH1
SCHEMBL7358973 0.70 HSP90AA1 (0.49) CA12CA2MMP2MMP9MMP8
Phosphonic Acid SCHEMBL27297809 0.69 KCNJ11 (0.39) KCNJ11NPC1RAB9AKDM4EG6PD
SCHEMBL27338316 0.68 ALDH1A1 (0.37) CA2ALDH1A1CYP3A4HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288065-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PARKINSON*S AND ALZHEIMER*S DISEASE SCHERING AKTIENGESEELLSCHAFT (DE) 2001-09-11 US disclosed
US-6057304-A Quinoxaline-phosphonic acid derivatives SCHERING AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed
CN-1038840-C para-dinitrogen naphthalene derivative, its preparation method and its medical use SCHERING AG (DE) 1998-06-24 CN disclosed
EP-0565683-A1 QUINOXALINE DERIVATES WITH AFFINITY FOR QUISQUALATE-RECEPTORS SCHERING AKTIENGESELLSCHAFT (DE) 1993-10-20 EP disclosed
CN-1072929-A Para-dinitronaphthalene derivative, preparation method and medical application thereof SCHERING AG (DE) 1993-06-09 CN disclosed
WO-1993008173-A1 QUINOXALINE DERIVATES WITH AFFINITY FOR QUISQUALATE-RECEPTORS SCHERING AKTIENGESELLSCHAFT (DE) 1993-04-29 WO disclosed