SCHEMBL8621279

SCHEMBL8621279

CC(C#N)Nc1c(N)ccc2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.36
HSD17B10 Q99714 3/20 0.36
TSHR P16473 3/20 0.36
HPGD P15428 2/20 0.36
CYP3A4 P08684 1/20 0.36
KEAP1 Q14145 1/20 0.36
HPRT1 P00492 2/20 0.35
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 2/20 0.34
MAPT P10636 2/20 0.34
KMT2A Q03164 2/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
CASP1 P29466 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
CASP7 P55210 1/20 0.34
CYP2A6 P11509 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27338316 0.83 ALDH1A1 (0.37) ALDH1A1HSD17B10TSHRHPGDCYP3A4
SCHEMBL8617883 0.79 ALDH1A1 (0.44) ALDH1A1TSHRCYP3A4HPRT1KDM4E
SCHEMBL8623600 0.78 NCEH1 (0.37) ALDH1A1HSD17B10TSHRHPGDCYP3A4
SCHEMBL6171290 0.78 MAPT (0.38) ALDH1A1HSD17B10HPGDKDM4EMEN1
SCHEMBL8620493 0.74 ALDH1A1 (0.38) ALDH1A1HSD17B10TSHRHPGDCYP3A4
SCHEMBL680370 0.74 AKR1B1 (0.40) ALDH1A1HSD17B10TSHRKDM4EMEN1
SCHEMBL7353058 0.73 CA12 (0.44) ALDH1A1HSD17B10TSHRHPGDCYP3A4
SCHEMBL21555507 0.72 ALDH1A1 (0.46) ALDH1A1HSD17B10TSHRHPGDCYP3A4
SCHEMBL23961077 0.68 CA1 (0.36) ALDH1A1HSD17B10HPGDHPRT1KDM4E
Acetonitrile SCHEMBL27651258 0.67 ALDH1A1 (0.45) ALDH1A1HSD17B10TSHRHPGDCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1041935-C Benzo[f]quinoxalindione derivatives, their preparation and their use in drugs SCHERING AG (DE) 1999-02-03 CN disclosed
US-5710138-A Benzo f!quinoxalinedione derivatives, their production and use in pharmaceutical agents SCHERING AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
EP-0696289-B1 BENZO[F]QUINOXALINDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN DRUGS SCHERING AG (DE) 1997-03-12 EP disclosed
CN-1122136-A Benzo[f]quinoxalindione derivatives, their preparation and their use in drugs SCHERING AG (DE) 1996-05-08 CN disclosed
EP-0696289-A1 BENZO F]QUINOXALINDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN DRUGS SCHERING AG (DE) 1996-02-14 EP disclosed
WO-1994025470-A1 BENZO[F]QUINOXALINDIONE DERIVATIVES, THEIR PREPARATION AND THEIR USE IN DRUGS SCHERING AKTIENGESELLSCHAFT (DE) 1994-11-10 WO disclosed