SCHEMBL7358973

SCHEMBL7358973

CC(Nc1ccc2ccccc2c1[N+](=O)[O-])P(=O)(O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.49
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49
TSHR P16473 1/20 0.49
NCEH1 Q6PIU2 1/20 0.45
CA12 O43570 1/20 0.43
CA2 P00918 1/20 0.43
MMP2 P08253 1/20 0.43
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
MMP14 P50281 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CYP3A4 P08684 1/20 0.43
MEN1 O00255 5/20 0.38
KMT2A Q03164 5/20 0.38
LMNA P02545 4/20 0.38
MAPT P10636 4/20 0.38
NPSR1 Q6W5P4 2/20 0.38
HTT P42858 2/20 0.38
FDPS P14324 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8622309 0.84 HSP90AA1 (0.42) HSP90AA1CRHBPCRHR2TSHRNCEH1
SCHEMBL8622301 0.82 HSP90AA1 (0.45) HSP90AA1CRHBPCRHR2TSHRNCEH1
SCHEMBL7358348 0.79 ALDH1A1 (0.43) TSHRNCEH1CA12CA2MMP2
SCHEMBL7360428 0.78 HSP90AA1 (0.48) HSP90AA1CRHBPCRHR2TSHRNCEH1
SCHEMBL7357998 0.78 CA12 (0.48) NCEH1CA12CA2MMP2MMP9
SCHEMBL8620563 0.77 HSP90AA1 (0.50) HSP90AA1CRHBPCRHR2TSHRNCEH1
SCHEMBL8622264 0.77 HSP90AA1 (0.41) HSP90AA1CRHBPCRHR2TSHRNCEH1
SCHEMBL4430656 0.77 CA12 (0.71) CA12CA2MMP2MMP9MMP8
SCHEMBL8620764 0.75 HSP90AA1 (0.39) HSP90AA1CRHBPCRHR2TSHRNCEH1
SCHEMBL8623634 0.75 HSP90AA1 (0.39) HSP90AA1CRHBPCRHR2TSHRNCEH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288065-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PARKINSON*S AND ALZHEIMER*S DISEASE SCHERING AKTIENGESEELLSCHAFT (DE) 2001-09-11 US disclosed
US-6057304-A Quinoxaline-phosphonic acid derivatives SCHERING AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed
CN-1038840-C para-dinitrogen naphthalene derivative, its preparation method and its medical use SCHERING AG (DE) 1998-06-24 CN disclosed
CN-1072929-A Para-dinitronaphthalene derivative, preparation method and medical application thereof SCHERING AG (DE) 1993-06-09 CN disclosed
WO-1993008173-A1 QUINOXALINE DERIVATES WITH AFFINITY FOR QUISQUALATE-RECEPTORS SCHERING AKTIENGESELLSCHAFT (DE) 1993-04-29 WO disclosed