SCHEMBL7354063

SCHEMBL7354063

CC1CC(=O)c2c(OC(N)=S)ccc(Br)c2C1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.40
CYP1A2 P05177 1/20 0.35
BRD4 O60885 2/20 0.34
ALDH1A1 P00352 1/20 0.31
PKM P14618 1/20 0.31
STAT3 P40763 1/20 0.30
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7354058 1.00 KDM4E (0.40) KDM4ECYP1A2BRD4ALDH1A1PKM
SCHEMBL7359720 0.80 KDM4E (0.62) KDM4ECYP1A2BRD4ALDH1A1ACHE
SCHEMBL7349576 0.76 KDM4E (0.40) KDM4EBRD4ALDH1A1
SCHEMBL7355336 0.75 GABRG2 (0.58) BRD4STAT3
SCHEMBL7350948 0.75 GABRG2 (0.58) BRD4STAT3
SCHEMBL7351763 0.74 STAT3 (0.44) KDM4ECYP1A2BRD4ALDH1A1STAT3
SCHEMBL7349414 0.72 GABRG2 (0.39) KDM4ECYP1A2STAT3
SCHEMBL7357100 0.68 KDM4E (0.35) KDM4EBRD4ALDH1A1PKMSTAT3
SCHEMBL10982867 0.67 ACHE (0.62) KDM4EBRD4ALDH1A1ACHE
SCHEMBL7361535 0.66 GABRG2 (0.58) KDM4EBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156761-A Substituted tetralone derivatives for enhancing cognition MERCK SHARPE & DOHME LIMITED (GB) 2000-12-05 US disclosed