SCHEMBL7354099

SCHEMBL7354099

COc1ccc(NC(=O)c2ccc(C(=O)N3CCCc4ccccc43)cc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.80
TSHR P16473 1/20 0.80
MAPT P10636 1/20 0.73
RAB9A P51151 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359695 0.90 AVPR1A (0.67)
SCHEMBL7350530 0.90 TSHR (0.77) ALDH1A1TSHRSMN1; SMN2
SCHEMBL7345982 0.89 RAB9A (0.78) RAB9A
SCHEMBL7347903 0.89 ALDH1A1 (0.75) ALDH1A1TSHRRAB9ASMN1; SMN2
SCHEMBL7350425 0.89 TSHR (0.71) ALDH1A1TSHR
SCHEMBL6971547 0.88 AVPR2 (0.76) ALDH1A1TSHRMAPT
SCHEMBL7347848 0.88 RAB9A (0.72) RAB9A
SCHEMBL7353560 0.87 TSHR (0.72) ALDH1A1TSHRSMN1; SMN2
SCHEMBL7348562 0.86 TSHR (0.70) ALDH1A1TSHRSMN1; SMN2
SCHEMBL7348778 0.85 AVPR1A (0.76) RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5985869-A USEFUL AS VASODILATORS, HYPOTENSIVE AGENTS, WATER DIURETICS, PLATELET AGGLUTINATION INHIBITORS OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1999-11-16 US disclosed
US-5753677-A Benzoheterocyclic compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed
US-5559230-A VASOPRESSIN ANTAGONISTS, QUINOLINES, BENZAZEPINES, VASODILATION, HYPOTENSIVE AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-09-24 US disclosed
EP-0450097-B1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMA CO LTD (JP) 1996-04-24 EP disclosed
WO-1991005549-A1 BENZOHETEROCYCLIC COMPOUNDS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-05-02 WO disclosed