SCHEMBL7354552

SCHEMBL7354552

O=S(=O)(Cl)c1cccc(S(=O)(=O)NCc2ccccc2)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.69
LMNA P02545 4/20 0.61
SLC12A2 P55011 1/20 0.61
SLC12A5 Q9H2X9 1/20 0.61
HDAC2 Q92769 2/20 0.59
HDAC8 Q9BY41 2/20 0.59
HDAC6 Q9UBN7 2/20 0.59
HTT P42858 1/20 0.59
CYP19A1 P11511 3/20 0.56
CA12 O43570 2/20 0.55
CA9 Q16790 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
ATM Q13315 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
VCAM1 P19320 1/20 0.55
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
ALDH1A1 P00352 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27670793 0.84 KEAP1 (0.69) KEAP1LMNASLC12A2SLC12A5HDAC2
SCHEMBL407414 0.82 KEAP1 (1.00) KEAP1LMNASLC12A2SLC12A5HDAC2
SCHEMBL14025561 0.82 KEAP1 (0.71) KEAP1LMNASLC12A2SLC12A5HDAC2
SCHEMBL29951672 0.81 KEAP1 (0.65) KEAP1LMNASLC12A2SLC12A5HDAC2
SCHEMBL2056065 0.81 KEAP1 (0.65) KEAP1LMNASLC12A2SLC12A5HDAC2
SCHEMBL21048461 0.81 KEAP1 (0.81) KEAP1LMNAHDAC2HDAC8HDAC6
Hydrochloric Acid SCHEMBL3516799 0.81 KEAP1 (0.96) KEAP1LMNASLC12A2SLC12A5HDAC2
SCHEMBL1858605 0.81 KEAP1 (0.69) KEAP1LMNASLC12A2SLC12A5HDAC2
SCHEMBL16660687 0.81 ALDH1A1 (0.73) KEAP1LMNASLC12A2SLC12A5HDAC2
SCHEMBL31339948 0.81 CYP19A1 (0.85) KEAP1LMNASLC12A2SLC12A5HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686486-A 4-hydroxy-benzopyran-2-ones and 4-hydroxy-cycloalkyl b!pyran-2-ones useful to treat retroviral infections PHARMACIA & UPJOHN COMPANY (US) 1997-11-11 US disclosed
EP-0682663-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS PHARMACIA & UPJOHN COMPANY (US) 1995-11-22 EP disclosed
WO-1994018188-A1 4-HYDROXY-BENZOPYRAN-2-ONES AND 4-HYDROXY-CYCLOALKYL[B]PYRAN-2-ONES USEFUL TO TREAT RETROVIRAL INFECTIONS THE UPJOHN COMPANY (US) 1994-08-18 WO disclosed