SCHEMBL7355420

SCHEMBL7355420

CC#CCOc1ccc(C(=S(=O)=O)C2(C(=O)NO)CCN(C(=O)c3cccs3)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 17/20 0.64
MMP2 P08253 11/20 0.64
MMP1 P03956 10/20 0.64
MMP14 P50281 9/20 0.64
ADAM17 P78536 17/20 0.52
MMP9 P14780 7/20 0.52
ALDH1A1 P00352 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6266377 0.85 ADAM17 (0.61) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL7356262 0.81 ADAM17 (0.59) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL7360886 0.81 ADAM17 (0.61) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL7363135 0.81 ADAM17 (0.51) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL7363196 0.80 ADAM17 (0.63) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL3944024 0.80 MMP13 (0.77) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL6265588 0.79 ADAM17 (0.49) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL3940450 0.78 MMP2 (1.00) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL7394688 0.76 ADAM17 (0.80) MMP13MMP2MMP1MMP14ADAM17
SCHEMBL6265492 0.75 MMP2 (0.92) MMP13MMP2MMP1MMP14ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147085-A1 ALKYNYL CONTAINING HYDROXAMIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MATRIX METALLOPROTEINASE (MMP) INHIBITORS / TNF-ALPHA CONVERTING ENZYME (TACE) INHIBITORS American Cyanamid Company (US) 2001-10-24 EP claimed
WO-2000044723-A1 ALKYNYL CONTAINING HYDROXAMIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MATRIX METALLOPROTEINASE (MMP) INHIBITORS/TNF-ALPHA CONVERTING ENZYME (TACE) INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-08-03 WO claimed