SCHEMBL7356262

SCHEMBL7356262

CC#CCOc1ccc(C(=S(=O)=O)C2(C(=O)NO)CCN(CC#CC)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADAM17 P78536 20/20 0.59
MMP13 P45452 16/20 0.59
MMP2 P08253 9/20 0.59
MMP1 P03956 9/20 0.48
MMP9 P14780 8/20 0.48
MMP14 P50281 7/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360886 0.92 ADAM17 (0.61) ADAM17MMP13MMP2MMP1MMP9
Hydrochloric Acid SCHEMBL7383902 0.89 MMP2 (0.79) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6266377 0.88 ADAM17 (0.61) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL7363135 0.84 ADAM17 (0.51) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL7363196 0.83 ADAM17 (0.63) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL7355420 0.81 MMP13 (0.64) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6265588 0.80 ADAM17 (0.49) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL7394688 0.79 ADAM17 (0.80) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6795694 0.75 MMP1 (0.59) ADAM17MMP13MMP2MMP1MMP9
SCHEMBL6267986 0.74 ADAM17 (1.00) ADAM17MMP13MMP2MMP1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147085-A1 ALKYNYL CONTAINING HYDROXAMIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MATRIX METALLOPROTEINASE (MMP) INHIBITORS / TNF-ALPHA CONVERTING ENZYME (TACE) INHIBITORS American Cyanamid Company (US) 2001-10-24 EP disclosed
WO-2000044723-A1 ALKYNYL CONTAINING HYDROXAMIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MATRIX METALLOPROTEINASE (MMP) INHIBITORS/TNF-ALPHA CONVERTING ENZYME (TACE) INHIBITORS AMERICAN CYANAMID COMPANY (US) 2000-08-03 WO disclosed