SCHEMBL7355965

SCHEMBL7355965

CC(C)(C)[Si](C)(C)OC(C(=O)c1ccncc1)c1ccc(F)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.43
ADRB2 P07550 2/20 0.38
ADRB1 P08588 2/20 0.38
ADRB3 P13945 2/20 0.38
CYP26A1 O43174 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
PTGS2 P35354 2/20 0.35
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MAPKAPK2 P49137 1/20 0.34
MEN1 O00255 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
MAPT P10636 1/20 0.34
KDM5A P29375 1/20 0.34
KDM4C Q9H3R0 1/20 0.34
KDM5B Q9UGL1 1/20 0.34
NPC1 O15118 1/20 0.34
USP2 O75604 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2660701 0.95 LTA4H (0.43) LTA4HADRB2ADRB1ADRB3CYP26A1
SCHEMBL2527651 0.84 ALDH1A1 (0.47) ADRB2ADRB1ADRB3L3MBTL1KMT2A
SCHEMBL7510812 0.84 EPHX2 (0.46) PTGS2
SCHEMBL8101790 0.83 CES2 (0.43) KMT2ANPC1RAB9AKDM4EALDH1A1
SCHEMBL8110660 0.82 CES2 (0.39) ADRB2ADRB1ADRB3KMT2AUSP2
SCHEMBL2659647 0.82 NPC1 (0.39) ADRB2ADRB1ADRB3KMT2APOLB
SCHEMBL8110197 0.81 CHRNA1 (0.47) ADRB2ADRB1ADRB3SMN1; SMN2RAB9A
SCHEMBL5482456 0.78 AKR1C3 (0.43) CYP26A1L3MBTL1PTGS2MAPT
SCHEMBL4024359 0.75 CES2 (0.44) LTA4HADRB2ADRB1ADRB3CYP26A1
SCHEMBL8111034 0.75 SLC6A2 (0.48) L3MBTL1KMT2APOLBSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995003297-A1 IMIDAZOLES FOR TREATING CYTOKINE MEDIATED DISEASE SMITHKLINE BEECHAM CORPORATION (US) 1995-02-02 WO disclosed
EP-0623126-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS CYTOKINE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-11-09 EP disclosed
WO-1993014081-A1 IMIDAZOLE DERIVATIVES AND THEIR USE AS CYTOKINE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1993-07-22 WO disclosed