SCHEMBL7356463

SCHEMBL7356463

CCOC(=O)CCN(C(=O)c1cccnc1)c1ccc2c(C(=O)CCc3ccc(C#N)cc3)cn(C)c2c1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITK Q08881 3/20 0.37
USP14 P54578 1/20 0.36
PDK1 Q15118 1/20 0.35
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 2/20 0.34
ELANE P08246 2/20 0.34
CACNA1H O95180 1/20 0.34
HTT P42858 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TXK P42681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352512 0.86 ITK (0.37) ITKUSP14PDK1KDM4EALDH1A1
Hydrochloric Acid SCHEMBL7362428 0.82 NQO2 (0.41)
Hydrochloric Acid SCHEMBL7357504 0.74 F2 (0.46) KDM4EALDH1A1MEN1HPGDKMT2A
Hydrochloric Acid SCHEMBL7360735 0.74 F2 (0.46)
SCHEMBL7362376 0.74 KMT2A (0.39) USP14KDM4EALDH1A1MEN1KMT2A
SCHEMBL7361404 0.74 USP14 (0.34) USP14MAPTELANECACNA1H
SCHEMBL6781674 0.73 F2 (0.48) ITKMAPTHTTHSD17B10
SCHEMBL7362439 0.72 LMNA (0.38) USP14KDM4EMAPTELANECACNA1H
Hydrochloric Acid SCHEMBL7350504 0.72 NQO2 (0.37) KDM4EALDH1A1MEN1HPGDKMT2A
Hydrochloric Acid SCHEMBL7352566 0.72 F2 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed