SCHEMBL7361404

SCHEMBL7361404

CCOC(=O)CCN(C(=O)Oc1ccc2c(c1)c(C(=O)CCc1ccc(C#N)cc1)cn2C)c1cccnn1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
USP14 P54578 2/20 0.34
CYP19A1 P11511 2/20 0.34
ELANE P08246 1/20 0.32
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HTR3E A5X5Y0 1/20 0.30
HTR3B O95264 1/20 0.30
HTR3A P46098 1/20 0.30
HTR3D Q70Z44 1/20 0.30
HTR3C Q8WXA8 1/20 0.30
CACNA1H O95180 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7362376 0.87 KMT2A (0.39) USP14CYP19A1MAPTTDP1
SCHEMBL7352796 0.85 GAA (0.35) USP14ELANEMAPTTDP1HTR3E
SCHEMBL7353094 0.84 ELANE (0.35) USP14CYP19A1ELANEMAPTTDP1
SCHEMBL7359804 0.84 SMN1; SMN2 (0.37) CYP19A1MAPTHTR3EHTR3BHTR3A
SCHEMBL7356973 0.81 USP14 (0.33) USP14CYP19A1ELANEMAPTTDP1
SCHEMBL7356649 0.81 USP14 (0.37) USP14CYP19A1MAPTTDP1CACNA1H
SCHEMBL7354323 0.81 USP14 (0.38) USP14CYP19A1MAPTTDP1CACNA1H
Hydrochloric Acid SCHEMBL7357014 0.80 NQO2 (0.48)
Hydrochloric Acid SCHEMBL7358291 0.79 F2 (0.37)
SCHEMBL7359771 0.79 PSMB5 (0.39) USP14CYP19A1MAPTTDP1CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed