SCHEMBL7356989

SCHEMBL7356989

CCOC(=O)Cc1c(C)[nH]c(=O)c([N+](=O)[O-])c1SCCO

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.41
KDM4E B2RXH2 4/20 0.39
MAPK1 P28482 2/20 0.38
ALDH1A1 P00352 4/20 0.37
HPGD P15428 2/20 0.37
HSD17B10 Q99714 2/20 0.37
SMN1; SMN2 Q16637 4/20 0.35
KMT2A Q03164 3/20 0.35
TDP1 Q9NUW8 1/20 0.35
LMNA P02545 3/20 0.34
MAPT P10636 4/20 0.34
MEN1 O00255 1/20 0.34
HTT P42858 1/20 0.34
CASP6 P55212 1/20 0.34
ATM Q13315 1/20 0.34
USP2 O75604 1/20 0.34
TSHR P16473 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357903 0.90 POLB (0.40) POLBKDM4EMAPK1ALDH1A1HPGD
SCHEMBL7362798 0.71 POLB (0.39) POLBKDM4EMAPK1ALDH1A1HPGD
SCHEMBL7012269 0.64 GRIN2D (0.48) POLBSMN1; SMN2KMT2AMAPTMEN1
SCHEMBL9268773 0.63 POLB (0.71) POLBKDM4EMAPK1ALDH1A1HPGD
SCHEMBL7356994 0.63 ALDH1A1 (0.42) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL9846189 0.63 GRIN2D (0.45) POLBKDM4EALDH1A1HPGDHSD17B10
SCHEMBL7454505 0.62 MAPK1 (0.46) POLBKDM4EMAPK1ALDH1A1HPGD
SCHEMBL5468196 0.62 LMNA (0.41) POLBKDM4EALDH1A1KMT2ALMNA
SCHEMBL30433473 0.62 POLB (0.66) POLBKDM4EMAPK1ALDH1A1HPGD
SCHEMBL3571118 0.61 ALDH1A1 (0.51) POLBKDM4EALDH1A1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1117660-A4 THROMBIN INHIBITORS MERCK & CO INC (US) 2002-01-09 EP disclosed
EP-1117660-A1 THROMBIN INHIBITORS Merck & Co., Inc. (US) 2001-07-25 EP disclosed
WO-2000018762-A1 THROMBIN INHIBITORS MERCK & CO., INC. (US) 2000-04-06 WO disclosed