SCHEMBL7357789

SCHEMBL7357789

CC(C)[C@H](N)C(=O)N(C(=O)Cc1ccc(-c2ccccc2)cc1)c1n[nH]c(=S)s1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA12 O43570 6/20 0.40
CA1 P00915 6/20 0.40
CA2 P00918 6/20 0.40
CA5A P35218 6/20 0.40
CA9 Q16790 6/20 0.40
CA5B Q9Y2D0 6/20 0.40
MMP3 P08254 7/20 0.39
ROCK2 O75116 2/20 0.35
ROCK1 Q13464 1/20 0.35
MMP1 P03956 2/20 0.35
MMP2 P08253 1/20 0.35
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7366460 0.83 MMP3 (0.42) MMP3MMP1MMP2
SCHEMBL7356789 0.71 MMP3 (0.43) MMP3MMP1MMP2
SCHEMBL7396119 0.69 MMP3 (0.44) MMP3MMP1MMP2
SCHEMBL7357793 0.66 MMP3 (0.54) MMP3MMP1MMP2ALDH1A1MAPT
SCHEMBL20904188 0.62 ABCC4 (0.55) CA12CA1CA2CA5ACA9
SCHEMBL2625190 0.61 LMNA (0.62) ALDH1A1MAPTHPGD
SCHEMBL20888587 0.61 LMNA (0.62) CA12CA1CA2CA5ACA9
SCHEMBL12261267 0.59 BACE1 (0.64) ALDH1A1
SCHEMBL10382329 0.59 BACE1 (0.64) ALDH1A1
SCHEMBL1751593 0.59 BACE1 (0.64) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998025949-A1 SUBSTITUTED 5-AMINO-1,3,4-THIADIAZOLE-2-THIONES PROSCRIPT, INC. (US) 1998-06-18 WO disclosed
EP-0845002-A2 AMINO ACID AMIDES OF 5-AMINO-1,3,4-THIADIAZONES AND THEIR USE AS INHIBITORS FOR MATRIX METALLOPROTEINASES PROSCRIPT, INC. (US) 1998-06-03 EP disclosed
US-5677282-A ENZYME INHIBITOR; OSTEOARTHRITIS AND RHEUMATIC DISORDERS PROSCRIPT, INC. (US) 1997-10-14 US disclosed
WO-1996040745-A2 AMINO ACID AMIDES OF 5-AMINO-1,3,4-THIADIAZONES AND THEIR USE AS INHIBITORS FOR MATRIX METALLOPROTEINASES PROSCRIPT, INC. (US) 1996-12-19 WO disclosed