SCHEMBL7358689

SCHEMBL7358689

N#Cc1ccc(NC(=O)Cn2ccc3cc(NS(=O)(=O)c4cccc5cccnc45)ccc32)cc1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NTSR1 P30989 3/20 0.67
PKLR P30613 4/20 0.51
ALDH1A1 P00352 2/20 0.47
GAA P10253 2/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
EGLN1 Q9GZT9 1/20 0.45
TP53 P04637 1/20 0.45
HTT P42858 1/20 0.45
FABP1 P07148 2/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
PKM P14618 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
RORC P51449 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3196667 0.80 NTSR1 (0.79) NTSR1PKLRALDH1A1GAAFABP1
SCHEMBL3185394 0.80 NTSR1 (1.00) NTSR1
SCHEMBL27650858 0.77 NTSR1 (0.62) NTSR1ALDH1A1GAAMEN1KMT2A
SCHEMBL3195492 0.76 NTSR1 (0.62) NTSR1PKLRALDH1A1GAAMEN1
SCHEMBL3146898 0.76 HTR6 (0.72) NTSR1ALDH1A1GAAMEN1KMT2A
SCHEMBL8026334 0.75 F2 (0.55) NTSR1PKLRALDH1A1GAAMEN1
SCHEMBL7357627 0.75 PKLR (0.46) NTSR1PKLRALDH1A1GAAMEN1
SCHEMBL6572882 0.75 MEN1 (0.52) PKLRALDH1A1GAAMEN1KMT2A
SCHEMBL6633872 0.75 F2 (0.50) NTSR1PKLRALDH1A1GAAMEN1
SCHEMBL8029757 0.74 F2 (0.55) PKLRALDH1A1GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed