SCHEMBL7358788

SCHEMBL7358788

Cc1nc2ccccc2c([O])c1C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.59
GPR3 P46089 1/20 0.57
HSD17B10 Q99714 2/20 0.52
ALDH1A1 P00352 2/20 0.52
CYP1A2 P05177 2/20 0.52
HPGD P15428 1/20 0.52
NUDT1 P36639 1/20 0.52
HTT P42858 2/20 0.50
MAPT P10636 2/20 0.47
TP53 P04637 1/20 0.47
ERN1 O75460 1/20 0.47
CASP3 P42574 1/20 0.47
ELANE P08246 1/20 0.44
PARP1 P09874 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPK1 P28482 1/20 0.44
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL231530 0.80 GPR3 (0.64) PDE10AGPR3HSD17B10ALDH1A1CYP1A2
SCHEMBL8061027 0.80 HSD17B10 (0.58) PDE10AGPR3HSD17B10ALDH1A1CYP1A2
Ammonia Solution, Strong SCHEMBL28822932 0.78 GPR3 (0.61) PDE10AGPR3HSD17B10ALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL27521191 0.78 GPR3 (0.61) PDE10AGPR3HSD17B10ALDH1A1CYP1A2
SCHEMBL4894495 0.77 KDM4E (0.56) GPR3HSD17B10ALDH1A1HPGDHTT
SCHEMBL27296318 0.77 ALDH1A1 (0.64) PDE10AGPR3HSD17B10ALDH1A1CYP1A2
SCHEMBL30025532 0.77 ALDH1A1 (0.64) PDE10AGPR3HSD17B10ALDH1A1CYP1A2
SCHEMBL6788479 0.75 GPR3 (0.57) PDE10AGPR3HSD17B10ALDH1A1CYP1A2
SCHEMBL11985944 0.75 GPR3 (0.57) PDE10AGPR3HSD17B10ALDH1A1CYP1A2
SCHEMBL6215008 0.75 GPR3 (0.57) PDE10AGPR3HSD17B10ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027332-A1 NOVEL LACTAM METALLOPROTEASE INHIBITORS Du Pont Pharmaceuticals Company (US) 2000-08-16 EP disclosed
US-6057336-A ANTIINFLAMMATORY AGENTS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2000-05-02 US disclosed
WO-1999018074-A1 NOVEL LACTAM METALLOPROTEASE INHIBITORS Britol-Myers Squibb Pharma Company (US) 1999-04-15 WO disclosed