SCHEMBL7358963

SCHEMBL7358963

O=C1CCC(c2ccc(CCO)cc2)=NN1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.58
MAPT P10636 2/20 0.52
LMNA P02545 2/20 0.52
NPY1R P25929 1/20 0.52
NPY2R P49146 1/20 0.52
PDE3B Q13370 13/20 0.52
PDE3A Q14432 12/20 0.52
KCNH2 Q12809 1/20 0.51
KMT2A Q03164 1/20 0.49
PDE4A P27815 5/20 0.48
PDE4B Q07343 5/20 0.48
PDE4C Q08493 5/20 0.48
PDE4D Q08499 5/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7312349 0.87 SMN1; SMN2 (0.62) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL21969533 0.84 MAPT (0.63) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL7297347 0.84 SMN1; SMN2 (0.58) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL10353452 0.83 SMN1; SMN2 (0.81) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL8114164 0.82 SMN1; SMN2 (0.55) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL8110737 0.81 SMN1; SMN2 (0.54) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL7298599 0.80 SMN1; SMN2 (0.61) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL9815919 0.80 LMNA (0.65) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL8100532 0.80 SMN1; SMN2 (0.53) SMN1; SMN2MAPTLMNANPY1RNPY2R
SCHEMBL8100411 0.80 SMN1; SMN2 (0.53) SMN1; SMN2MAPTLMNANPY1RNPY2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4876255-A CARDIOVASCULAR BAYER AKTIENGESELLSCHAFT (DE) 1989-10-24 US disclosed
EP-0287866-A1 Substituted 1,4-dihydropyridines, method for their preparation and their use BAYER AG (DE) 1988-10-26 EP disclosed