SCHEMBL7359093

SCHEMBL7359093

CC(C)(C)OC(=O)Cn1c(=O)c(=O)[nH]c2cc(C(F)(F)F)ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.47
PDE9A O76083 2/20 0.47
GRIA1 P42261 8/20 0.45
GRIA2 P42262 8/20 0.45
GRIA3 P42263 8/20 0.45
GRIA4 P48058 8/20 0.45
GRIN1 Q05586 3/20 0.43
GRIN2B Q13224 3/20 0.43
GRIN2D O15399 2/20 0.43
GRIN3B O60391 2/20 0.43
GRIN2A Q12879 2/20 0.43
GRIN2C Q14957 2/20 0.43
GRIN3A Q8TCU5 2/20 0.43
GRIK1 P39086 3/20 0.42
GRIK2 Q13002 3/20 0.42
GRIK3 Q13003 3/20 0.42
GRIK4 Q16099 3/20 0.42
GRIK5 Q16478 3/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7486477 0.86 GRIA1 (0.58) PDE5APDE9AGRIA1GRIA2GRIA3
SCHEMBL7359701 0.83 GRIA1 (0.58) PDE5APDE9AGRIA1GRIA2GRIA3
SCHEMBL5551602 0.81 KDM4E (0.52) GRIA1GRIA2GRIA3GRIA4GRIN1
SCHEMBL9544064 0.79 GRIA1 (0.55) PDE5APDE9AGRIA1GRIA2GRIA3
SCHEMBL9613772 0.79 GRIA1 (0.66) GRIA1GRIA2GRIA3GRIA4GRIN1
SCHEMBL8611656 0.78 GRIK1 (0.52) PDE5APDE9AGRIA1GRIA2GRIA3
SCHEMBL8117343 0.77 MEN1 (0.47) PDE5APDE9AGRIA1GRIA2GRIA3
SCHEMBL7478166 0.77 PDE5A (0.50) PDE5APDE9AGRIA1GRIA2GRIA3
SCHEMBL24335140 0.75 PDE5A (0.48) PDE5APDE9AGRIA1GRIA2GRIA3
SCHEMBL29580737 0.75 PDE5A (0.48) PDE5APDE9AGRIA1GRIA2GRIA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288065-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PARKINSON*S AND ALZHEIMER*S DISEASE SCHERING AKTIENGESEELLSCHAFT (DE) 2001-09-11 US disclosed
US-6057304-A Quinoxaline-phosphonic acid derivatives SCHERING AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed