SCHEMBL7359102

SCHEMBL7359102

COC(=O)C1CCC1C(O)C(N)Cc1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 6/20 0.52
CYP3A4 P08684 5/20 0.52
TSHR P16473 5/20 0.52
CYP2D6 P10635 2/20 0.52
HSD17B10 Q99714 2/20 0.52
MAPK1 P28482 1/20 0.52
CPB1 P15086 1/20 0.46
CYP2C19 P33261 6/20 0.45
CYP2C9 P11712 6/20 0.45
ALDH1A1 P00352 3/20 0.45
POLB P06746 1/20 0.45
LTA4H P09960 1/20 0.44
ANPEP P15144 3/20 0.42
LMNA P02545 3/20 0.42
LAP3 P28838 2/20 0.41
RNPEP Q9H4A4 1/20 0.41
DNPEP Q9ULA0 1/20 0.41
SLC15A1 P46059 1/20 0.41
MAPT P10636 1/20 0.41
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10590665 0.93 CYP3A4 (0.47) CYP1A2CYP3A4TSHRCYP2D6HSD17B10
SCHEMBL7361302 0.93 CYP1A2 (0.47) CYP1A2CYP3A4TSHRCYP2D6HSD17B10
SCHEMBL7357914 0.81 ESR1 (0.39) CYP1A2CYP3A4TSHRCYP2D6HSD17B10
SCHEMBL7360306 0.78 SLC15A1 (0.47) CYP1A2CYP3A4TSHRCYP2D6HSD17B10
SCHEMBL10591375 0.77 SLC15A1 (0.43) LTA4HANPEPLAP3RNPEPDNPEP
SCHEMBL7368172 0.77 TAAR1 (0.44) LTA4HANPEPLAP3RNPEPDNPEP
SCHEMBL7325758 0.72 KLK5 (0.58) KMT2A
SCHEMBL10377216 0.72 KLK5 (0.58) KMT2A
SCHEMBL11998024 0.71 CSNK1E (0.39) CYP2D6LTA4HANPEPLAP3RNPEP
SCHEMBL8174333 0.70 LTA4H (0.77) HSD17B10CYP2C19CYP2C9ALDH1A1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415981-A4 RETROVIRAL PROTEASE INHIBITORS 1991-10-09 EP disclosed
EP-0415981-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
EP-0342541-A2 Retroviral protease inhibitors ABBOTT LABORATORIES (US) 1989-11-23 EP disclosed
WO-1989010752-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed