SCHEMBL7359403

SCHEMBL7359403

NC(=O)C(=O)NCCc1ccc(O)c(OC(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOX4 Q9NPH5 1/20 0.47
ALDH1A1 P00352 7/20 0.44
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
PTGS1 P23219 1/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
EGFR P00533 1/20 0.43
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359573 0.91 ALDH1A1 (0.43) ALDH1A1KDM4ELMNAMAPTHPGD
SCHEMBL6811090 0.91 ALDH1A1 (0.47) ALDH1A1LMNAMAPTCA1CA2
SCHEMBL7359851 0.87 ALDH1A1 (0.56) ALDH1A1LMNAMAPTCA1CA2
SCHEMBL7362562 0.86 ALDH1A1 (0.58) ALDH1A1LMNAMAPTCA1CA2
SCHEMBL9275919 0.81 PDE4D (0.53) ALDH1A1
SCHEMBL7361910 0.80 MAPT (0.66) NOX4ALDH1A1KDM4ELMNAMAPT
SCHEMBL7358841 0.76 CA12 (0.69) ALDH1A1LMNAMAPTCA1CA2
SCHEMBL2746659 0.75 MTNR1A (0.61) NOX4ALDH1A1LMNAMTNR1AMTNR1B
SCHEMBL7348827 0.74 PDE4D (0.52)
SCHEMBL9269689 0.73 KMT2A (0.59) ALDH1A1LMNAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0538384-A4 OXAMIDES SMITHKLINE BEECHAM CORP (US) 1995-04-12 EP disclosed
US-5393788-A Phenylalkyl oxamides SMITHKLINE BEECHAM CORPORATION (US) 1995-02-28 US disclosed
EP-0538384-A1 OXAMIDES SMITHKLINE BEECHAM CORPORATION (US) 1993-04-28 EP disclosed
CN-1060652-A OXAMIDES SMITHKLINE BEECHAM CORP (US) 1992-04-29 CN disclosed
WO-1992000968-A1 OXAMIDES SMITHKLINE BEECHAM CORPORATION (US) 1992-01-23 WO disclosed