SCHEMBL6811090

SCHEMBL6811090

NC(=O)C(=O)NCCc1ccc(OC(F)F)c(OC(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA9 Q16790 1/20 0.46
THRB P10828 1/20 0.45
KMT2A Q03164 2/20 0.45
PLAAT3 P53816 1/20 0.44
PLAAT5 Q96KN8 1/20 0.44
PLAAT2 Q9NWW9 1/20 0.44
PLAAT4 Q9UL19 1/20 0.44
POLB P06746 3/20 0.44
MAPT P10636 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7359851 0.94 ALDH1A1 (0.56) ALDH1A1CA12CA1CA2CA9
SCHEMBL7362562 0.92 ALDH1A1 (0.58) ALDH1A1CA12CA1CA2CA9
SCHEMBL7359403 0.91 NOX4 (0.47) ALDH1A1CA12CA1CA2CA9
SCHEMBL7359573 0.90 ALDH1A1 (0.43) ALDH1A1CA12CA1CA2CA9
SCHEMBL9275919 0.87 PDE4D (0.53) ALDH1A1KMT2AMEN1PDE4APDE4B
SCHEMBL7358841 0.80 CA12 (0.69) ALDH1A1CA12CA1CA2CA9
SCHEMBL7348827 0.80 PDE4D (0.52) PDE4APDE4BPDE4CPDE4D
SCHEMBL9269689 0.77 KMT2A (0.59) ALDH1A1KMT2AMAPTMEN1LMNA
SCHEMBL7364544 0.74 ALDH1A1 (0.57) ALDH1A1KMT2APLAAT3PLAAT5PLAAT2
SCHEMBL7417119 0.73 PDE4B (0.61) PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5393788-A Phenylalkyl oxamides SMITHKLINE BEECHAM CORPORATION (US) 1995-02-28 US claimed
EP-1466598-A2 PDE-IV inhibitors SMITHKLINE BEECHAM CORPORATION (US) 2004-10-13 EP disclosed
EP-0710109-B1 Method for identifying a PDE IV inhibitor SMITHKLINE BEECHAM CORP (US) 2004-09-15 EP disclosed
US-5393788-A Phenylalkyl oxamides SMITHKLINE BEECHAM CORPORATION (US) 1995-02-28 US disclosed