SCHEMBL7359804

SCHEMBL7359804

COC(=O)CCN(C(=O)Oc1ccc2c(c1)c(C(=O)CCc1ccc(C#N)cc1)cn2C)c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.37
HSD17B10 Q99714 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 2/20 0.36
GAA P10253 2/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.34
MAPT P10636 1/20 0.34
CYP19A1 P11511 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
HAT1 O14929 2/20 0.32
EP300 Q09472 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7352796 0.88 GAA (0.35) SMN1; SMN2ALDH1A1MAPK1GAAL3MBTL1
SCHEMBL7361404 0.84 USP14 (0.34) MAPTCYP19A1HTR3EHTR3BHTR3A
SCHEMBL7362376 0.83 KMT2A (0.39) SMN1; SMN2ALDH1A1MEN1KMT2AMAPT
Hydrochloric Acid SCHEMBL7358962 0.82 F2 (0.46) FFAR1FFAR4
SCHEMBL7353094 0.82 ELANE (0.35) ALDH1A1MAPK1L3MBTL1MEN1KMT2A
Hydrochloric Acid SCHEMBL7357014 0.81 NQO2 (0.48)
SCHEMBL7356973 0.79 USP14 (0.33) MAPTCYP19A1HTR3EHTR3BHTR3A
Hydrochloric Acid SCHEMBL7361001 0.78 F2 (0.44) POLBFFAR1FFAR4
Iodide SCHEMBL7351241 0.77 NQO2 (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7358416 0.77 PLA2G4A (0.38) HSD17B10ALDH1A1CYP19A1FFAR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999028297-A1 SUBSTITUTED INDOLES, HAVING A THROMBIN INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-06-10 WO disclosed