SCHEMBL7360040

SCHEMBL7360040

COc1ccc(CCC2COC(c3ccccc3)O2)cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.49
KDM1A O60341 3/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
HIF1A Q16665 1/20 0.44
EPAS1 Q99814 1/20 0.44
EBP Q15125 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
TMEM97 Q5BJF2 1/20 0.42
ALDH1A1 P00352 2/20 0.41
POLB P06746 1/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
HTR2B P41595 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ATM Q13315 1/20 0.41
ABCB1 P08183 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
DRD4 P21917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10034619 0.83 ATM (0.54) SIGMAR1POLBKDM4EATM
SCHEMBL10695511 0.74 ATM (0.51) ADRA1AEBPSIGMAR1TMEM97POLB
SCHEMBL13381209 0.72 ADRA1A (0.46) ADRA1AALDH1A1MEN1KMT2A
SCHEMBL118949 0.71 ADRA1A (0.51) ADRA1AALDH1A1TDP1MEN1KMT2A
SCHEMBL9549492 0.71 ADRA1A (0.51) ADRA1AALDH1A1TDP1MEN1KMT2A
SCHEMBL1261811 0.71 CA2 (0.55) SIGMAR1ALDH1A1KDM4EATMSMN1; SMN2
SCHEMBL2689229 0.70 SLC6A4 (0.64) KDM4EATM
SCHEMBL2689969 0.70 SLC6A4 (0.64) KDM4EATM
SCHEMBL7978011 0.70 GRM2 (0.44) ADRA1AALDH1A1
SCHEMBL4924677 0.70 ADRA1A (0.43) ADRA1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0649426-A1 INHIBITORS OF RETROVIRAL PROTEASES HOECHST AKTIENGESELLSCHAFT (DE) 1995-04-26 EP claimed
WO-1994000461-A1 INHIBITORS OF RETROVIRAL PROTEASES HOECHST AKTIENGESELLSCHAFT (DE) 1994-01-06 WO claimed
EP-0435059-A1 Retroviral protease inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1991-07-03 EP claimed
EP-0428849-A2 Retroviral protease inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1991-05-29 EP claimed
EP-0649426-A1 INHIBITORS OF RETROVIRAL PROTEASES HOECHST AKTIENGESELLSCHAFT (DE) 1995-04-26 EP disclosed
WO-1994000461-A1 INHIBITORS OF RETROVIRAL PROTEASES HOECHST AKTIENGESELLSCHAFT (DE) 1994-01-06 WO disclosed
EP-0428849-A2 Retroviral protease inhibitors HOECHST AKTIENGESELLSCHAFT (DE) 1991-05-29 EP disclosed