SCHEMBL7360171

SCHEMBL7360171

COC(=O)COc1ccc(N2CCNCC2)cc1OCC(=O)OC

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 4/20 0.43
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
HTR1A P08908 2/20 0.43
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
IGF1R P08069 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
ALK Q9UM73 3/20 0.42
RAB9A P51151 1/20 0.41
LMNA P02545 1/20 0.41
HTR7 P34969 1/20 0.41
APP P05067 1/20 0.41
LRRK2 Q5S007 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1107020 0.95 CHRNB2 (0.46) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL1107049 0.90 ADRB1 (0.51) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL1107015 0.89 CHRNB2 (0.45) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL16788139 0.88 PTGDR (0.47) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL1107022 0.88 KMT2A (0.50) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL1107055 0.87 HTR6 (0.43) ADRB1HTR3EHTR3BHTR3AHTR3D
SCHEMBL1107056 0.86 HTR7 (0.51) ADRB1HTR1AHTR7LRRK2
SCHEMBL1115184 0.86 PTGDR (0.47) ADRB1ALKRAB9A
SCHEMBL1106993 0.86 HTR6 (0.49) ALK
SCHEMBL1107065 0.86 PTGDR (0.49) ADRB1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994356-A ANTICOAGULANT KARL THOMAE (DE) 1999-11-30 US disclosed
EP-0892783-A1 CARBOXYLIC ACID DERIVATIVES WITH AN AGGREGATION-INHIBITING ACTION Dr. Karl Thomae GmbH (DE) 1999-01-27 EP disclosed
WO-1997037975-A1 CARBOXYLIC ACID DERIVATIVES WITH AN AGGREGATION-INHIBITING ACTION DR. KARL THOMAE GMBH (DE) 1997-10-16 WO disclosed