SCHEMBL7360299

SCHEMBL7360299

CCCc1n[nH]c2c(=O)[nH]c(Cc3sccc3OCC)nc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 12/20 0.39
PDE1A P54750 6/20 0.37
PDE1B Q01064 6/20 0.37
PDE1C Q14123 6/20 0.37
KMT2A Q03164 3/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
PNP P00491 1/20 0.37
KDM4E B2RXH2 1/20 0.33
PDE6C P51160 3/20 0.32
PDE10A Q9Y233 2/20 0.31
PDE9A O76083 2/20 0.31
PDE3A Q14432 2/20 0.31
PDE2A O00408 1/20 0.31
ABCC4 O15439 1/20 0.31
ABCC5 O15440 1/20 0.31
PDE6D O43924 1/20 0.31
PDE8A O60658 1/20 0.31
ABCB11 O95342 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16972452 0.81 PDE1A (0.48) PDE5APDE1APDE1BPDE1CKMT2A
SCHEMBL6365530 0.76 PDE1A (0.46) PDE5APDE1APDE1BPDE1CKMT2A
SCHEMBL1028 0.74 PDE5A (0.68) PDE5APDE1APDE1BPDE1CKMT2A
SCHEMBL16972445 0.73 CCNB2 (0.41) KMT2AALDH1A1KDM4E
SCHEMBL7085453 0.72 PDE5A (0.36) PDE5APDE1APDE1BPDE1CKMT2A
SCHEMBL7019558 0.72 PARP1 (0.41) PDE5APDE1APDE1BPDE1CKMT2A
SCHEMBL3671939 0.72 PDE5A (0.55) PDE5APDE1APDE1BPDE1CPDE6C
SCHEMBL7431615 0.72 PDE5A (0.48) PDE5APDE1APDE1BPDE1CPDE6C
SCHEMBL7360293 0.71 ALDH1A1 (0.39) PDE5APDE1APDE1BPDE1CKMT2A
SCHEMBL8237549 0.70 CCNE2 (0.35) PDE5APDE1APDE1BPDE1CKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001003644-A9 PYRAZOLOPYRIMIDINONE DERIVATIVES CONJUGATED TO THIOPHENE MOIETIES OR BENZO [FUSED] 5-MEMBERED HETEROCYCLES FOR ERECTILE DYSFUNCTION PICOWER INST MED RES (US) 2001-11-29 WO disclosed