SCHEMBL7360293

SCHEMBL7360293

CCCc1n[nH]c2c(=O)n(C)c(-c3sccc3OCC)nc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
KDM4E B2RXH2 6/20 0.39
HPGD P15428 4/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
PDE5A O76074 13/20 0.37
PDE1A P54750 5/20 0.37
PDE1B Q01064 5/20 0.37
PDE1C Q14123 5/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
PDE6C P51160 3/20 0.35
GAA P10253 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
PDE3A Q14432 2/20 0.34
PDE2A O00408 1/20 0.34
ABCC4 O15439 1/20 0.34
ABCC5 O15440 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7446947 0.74 ALDH1A1 (0.46) ALDH1A1KDM4EHPGDCYP1A2PDE5A
SCHEMBL7019550 0.73 PDE5A (0.46) PDE5APDE1APDE1BPDE1CKMT2A
SCHEMBL3671938 0.73 PDE5A (0.63) PDE5APDE1APDE1BPDE1CPDE6C
SCHEMBL6249380 0.73 PDE5A (0.42) ALDH1A1KDM4EHPGDPDE5APDE1A
SCHEMBL7964905 0.72 PDE5A (0.38) ALDH1A1KDM4EHPGDPDE5APDE1A
SCHEMBL7360299 0.71 PDE5A (0.39) ALDH1A1KDM4EHPGDPDE5APDE1A
SCHEMBL14685954 0.70 KDM4E (0.48) KDM4EPDE5APDE1AKMT2APDE6C
SCHEMBL7428886 0.69 PDE5A (0.68) ALDH1A1KDM4EHPGDPDE5APDE1A
SCHEMBL7778185 0.69 PDE5A (0.54) PDE5APDE1APDE1BPDE1CPDE6C
SCHEMBL5085819 0.69 PDE5A (0.65) ALDH1A1PDE5AKMT2AMEN1PDE6C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001003644-A9 PYRAZOLOPYRIMIDINONE DERIVATIVES CONJUGATED TO THIOPHENE MOIETIES OR BENZO [FUSED] 5-MEMBERED HETEROCYCLES FOR ERECTILE DYSFUNCTION PICOWER INST MED RES (US) 2001-11-29 WO disclosed