SCHEMBL7360304

SCHEMBL7360304

C=C(c1ccc([N+](=O)[O-])cc1)C(N)c1cccc(C#N)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.41
KCNH2 Q12809 1/20 0.41
MAP2K1 Q02750 4/20 0.41
P4HB P07237 1/20 0.41
MAPT P10636 2/20 0.39
THRB P10828 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
ABCG2 Q9UNQ0 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HSP90AA1 P07900 1/20 0.39
OPRK1 P41145 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
VCAM1 P19320 1/20 0.38
FBP1 P09467 3/20 0.37
TSHR P16473 1/20 0.37
GRM4 Q14833 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7363757 0.75 KCNJ1 (0.51) KCNJ1KCNH2P4HBVCAM1FBP1
SCHEMBL7364292 0.71 KCNH2 (0.53) KCNJ1KCNH2P4HBABCG2ALDH1A1
SCHEMBL7363755 0.70 KCNJ1 (0.54) KCNJ1KCNH2P4HBABCG2VCAM1
SCHEMBL18920505 0.70 GRM4 (0.54) MEN1KMT2AALDH1A1GRM4
SCHEMBL6390843 0.70 TNF (0.52) MAPTMEN1KMT2AALDH1A1GRM4
SCHEMBL18116486 0.70 GRM4 (0.54) MEN1KMT2AALDH1A1GRM4
SCHEMBL27849068 0.70 GRM4 (0.54) MEN1KMT2AALDH1A1GRM4
SCHEMBL29913891 0.69 VCAM1 (0.64) KCNJ1KCNH2MAPTKMT2AALDH1A1
SCHEMBL57152 0.69 VCAM1 (0.64) KCNJ1KCNH2MAPTKMT2AALDH1A1
4-Nitrotoluene SCHEMBL15633856 0.68 ACHE (0.60) KCNJ1KCNH2MEN1KMT2AABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5942544-A α-branched anilines, toluenes, and analogs thereof as factor Xa inhibitors DUPONT PHARMACEUTICALS COMPANY (US) 1999-08-24 US disclosed
EP-0892780-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1999-01-27 EP disclosed
WO-1997030971-A1 M-AMIDINO PHENYL ANALOGS AS FACTOR Xa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-08-28 WO disclosed