SCHEMBL7360342

SCHEMBL7360342

NC(=O)c1ccccc1-c1ccc(Cl)cn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.51
CSNK1A1 P48729 1/20 0.45
TYRO3 Q06418 1/20 0.45
DYRK1B Q9Y463 1/20 0.45
ALOX5AP P20292 1/20 0.45
FEN1 P39748 1/20 0.45
PARP1 P09874 1/20 0.45
DHODH Q02127 1/20 0.43
RAB9A P51151 4/20 0.42
GRM5 P41594 1/20 0.42
NPC1 O15118 2/20 0.41
ALOX15 P16050 1/20 0.41
HTT P42858 1/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 2/20 0.41
CTSA P10619 1/20 0.41
NUDT1 P36639 1/20 0.40
MAPK9 P45984 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27909833 0.85 KDM4E (0.46) CSNK1A1DYRK1BPARP1DHODHRAB9A
SCHEMBL15903099 0.81 DHODH (0.44) BCAT2PARP1DHODHRAB9AGRM5
SCHEMBL1967459 0.81 BCAT2 (0.51) BCAT2CSNK1A1TYRO3DYRK1BALOX5AP
SCHEMBL3529606 0.81 BCAT2 (0.51) BCAT2CSNK1A1TYRO3DYRK1BALOX5AP
SCHEMBL27684371 0.81 BCAT2 (0.51) BCAT2CSNK1A1TYRO3DYRK1BALOX5AP
SCHEMBL4675603 0.78 RAB9A (0.40) DHODHRAB9ASMN1; SMN2
SCHEMBL197002 0.78 BCAT2 (0.71) BCAT2PARP1MAPTTDP1KDM4E
SCHEMBL25093211 0.77 BCAT2 (0.47) BCAT2CSNK1A1TYRO3DYRK1BALOX5AP
SCHEMBL30810258 0.77 KMT2A (0.54) BCAT2CSNK1A1TYRO3DYRK1BALOX5AP
SCHEMBL17894102 0.77 KMT2A (0.54) BCAT2CSNK1A1TYRO3DYRK1BALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023061440-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI), INC. (CN) 2023-04-20 WO disclosed
EP-4157888-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS Cullgen (Shanghai), Inc. (CN) 2023-04-05 EP disclosed
WO-2021239117-A1 MODIFIED PROTEINS AND PROTEIN DEGRADERS CULLGEN (SHANGHAI) , INC. (CN) 2021-12-02 WO disclosed
CN-105254623-A SUBSTITUTED BENZAMIDES HOFFMANN LA ROCHE 2016-01-20 CN disclosed
CN-102686563-A Substituted benzamide derivatives HOFFMANN LA ROCHE 2012-09-19 CN disclosed
EP-1140903-A1 AROMATIC AMIDES ELI LILLY AND COMPANY (US) 2001-10-10 EP disclosed
WO-2000039118-A1 AROMATIC AMIDES ELI LILLY AND COMPANY (US) 2000-07-06 WO disclosed