SCHEMBL7360933

SCHEMBL7360933

O=C(CNCC(=O)OC(=O)[C@@H]1CCCN1)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.48
HTR2B P41595 1/20 0.48
TSHR P16473 2/20 0.46
GLA P06280 1/20 0.46
CTSC P53634 1/20 0.42
ALDH1A1 P00352 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
MAPK1 P28482 1/20 0.40
GAA P10253 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ELANE P08246 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PREP P48147 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2228391 0.87 ALDH1A1 (0.55) HTR2CHTR2BTSHRCTSCALDH1A1
SCHEMBL23630151 0.84 ALDH1A1 (0.56) HTR2CHTR2BTSHRALDH1A1MAPK1
SCHEMBL4758450 0.83 TSHR (0.51) HTR2CHTR2BTSHRGLACTSC
SCHEMBL3447413 0.83 TSHR (0.51) HTR2CHTR2BTSHRGLACTSC
SCHEMBL489770 0.83 TSHR (0.51) HTR2CHTR2BTSHRGLACTSC
SCHEMBL4069956 0.82 TSHR (0.63) HTR2CHTR2BTSHRGLACTSC
SCHEMBL630517 0.82 TSHR (0.63) HTR2CHTR2BTSHRGLACTSC
SCHEMBL693351 0.82 TSHR (0.63) HTR2CHTR2BTSHRGLACTSC
SCHEMBL8134913 0.82 HTR2C (0.63) HTR2CHTR2BTSHRGLACTSC
SCHEMBL8773302 0.82 HTR2C (0.63) HTR2CHTR2BTSHRGLACTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4514391-A HYPOTENSIVE AGENTS; ANALGESICS E. R. SQUIBB & SONS, INC. (US) 1985-04-30 US disclosed
EP-0132304-A2 Hydroxy substituted peptide compounds E.R. Squibb & Sons, Inc. (US) 1985-01-30 EP disclosed