SCHEMBL7361786

SCHEMBL7361786

CCCCCNNC1=Nc2ccccc2C(c2ccccc2)=NC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.38
GABRA1 P14867 2/20 0.36
GABRG2 P18507 2/20 0.36
GABRB3 P28472 2/20 0.36
GABRA5 P31644 2/20 0.36
GABRA3 P34903 2/20 0.36
GABRA2 P47869 2/20 0.36
GABRB2 P47870 2/20 0.36
SOAT1 P35610 2/20 0.34
CCKBR P32239 1/20 0.34
HDAC3 O15379 2/20 0.33
HDAC1 Q13547 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
STAT1 P42224 1/20 0.33
RAB9A P51151 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11633602 0.87 OPRK1 (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7312843 0.76 IDO1 (0.47) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL11382448 0.74 IDO1 (0.47) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL11633599 0.71 L3MBTL1 (0.44) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7307919 0.71 GABRA1 (0.43) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL11639498 0.71 KMT2A (0.41) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL11788039 0.70 NPC1 (0.48) HDAC3HDAC1HDAC8NPC1ALDH1A1
SCHEMBL11633991 0.67 NPSR1 (0.44) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL11084408 0.67 IDO1 (0.49) IDO1GABRA1GABRG2GABRB3GABRA5
SCHEMBL10469905 0.66 IDO1 (0.51) IDO1GABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3987052-A SEDATIVES, TRANQUILIZERS, MUSCLE RELAXANTS THE UPJOHN COMPANY (US) 1976-10-19 US disclosed