SCHEMBL7362253

SCHEMBL7362253

CC(C)C[C@H](N)[C@@H](O)CCSCCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C19 P33261 1/20 0.45
CSNK1E P49674 1/20 0.41
ERAP1 Q9NZ08 4/20 0.40
ERAP2 Q6P179 3/20 0.40
IL1RN P18510 2/20 0.40
ANPEP P15144 4/20 0.37
LAP3 P28838 3/20 0.37
RNPEP Q9H4A4 2/20 0.37
DNPEP Q9ULA0 2/20 0.37
CA2 P00918 1/20 0.37
METAP2 P50579 2/20 0.36
AOC3 Q16853 1/20 0.36
METAP1 P53582 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
TAAR1 Q96RJ0 2/20 0.36
MAOA P21397 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8270986 0.86 ERAP1 (0.47) CSNK1EERAP1ERAP2IL1RNANPEP
SCHEMBL3506697 0.86 ERAP1 (0.47) CSNK1EERAP1ERAP2IL1RNANPEP
Hydrochloric Acid SCHEMBL7435119 0.84 ERAP1 (0.46) CSNK1EERAP1ERAP2IL1RNANPEP
SCHEMBL7439984 0.80 CA2 (0.42) CYP1A2CYP2D6CYP2C19CSNK1EERAP1
Hydrochloric Acid SCHEMBL10728209 0.79 CA2 (0.41) CSNK1EERAP1ERAP2IL1RNCA2
SCHEMBL9833212 0.79 ANPEP (0.40) CYP2D6ANPEPRNPEPDNPEP
SCHEMBL10975968 0.77 CYP1A2 (0.55) CYP1A2CYP2D6CYP2C19CA2AOC3
SCHEMBL7362251 0.77 ERAP1 (0.42) CYP1A2CYP2D6CYP2C19CSNK1EERAP1
SCHEMBL7396180 0.76 CA2 (0.44) CYP1A2CYP2C19CSNK1EERAP1ERAP2
SCHEMBL7396177 0.76 CA2 (0.44) CYP1A2CYP2C19CSNK1EERAP1ERAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415981-A4 RETROVIRAL PROTEASE INHIBITORS 1991-10-09 EP disclosed
EP-0415981-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1991-03-13 EP disclosed
EP-0258289-A4 PEPTIDE ANALOGS 1991-01-02 EP disclosed
EP-0342541-A2 Retroviral protease inhibitors ABBOTT LABORATORIES (US) 1989-11-23 EP disclosed
WO-1989010752-A1 RETROVIRAL PROTEASE INHIBITORS ABBOTT LABORATORIES (US) 1989-11-16 WO disclosed
US-4857507-A HYPOTENSIVE AGENT ABBOTT LABORATORIES (US) 1989-08-15 US disclosed
EP-0258289-A1 PEPTIDE ANALOGS ABBOTT LABORATORIES (US) 1988-03-09 EP disclosed
WO-1987004349-A1 PEPTIDE ANALOGS DELLARIA JOSEPH 1987-07-30 WO disclosed